Basic Peptide Information

DICL ID
DICL_Pep_02452
Ion Channel
Sodium channel type 5 subunit alpha
Peptide Function
Inhibitor
Gene Name
Scn5a

Activity Data (nM)

IC50
11.4 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
VRDGYIAQPENCVYHCFPGSSGCDTLCKEKGGTSGHCGFKVGHGLACWCNALPDNVGIIVEGEKCHS
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
α-toxin LqhIII
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
Not available

Experimental Conditions

pH
pH 7.4
Holding Potential (mV)
−120 mV
Temperature
21−24 °C
Test Method
Patch-clamping
Test Species
Not specified

Binding Information

Binding Site
Extracellular domain
Binding Site Residue
S1-S2 and S3-S4 linker

Ion Channel Information

Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available